Methimazole

  • Brand Name : Tapazole
  • Drug Class : Antithyroid Agents
  • Medical Author : John P. Cunha, DO, FACOEP
  • Medical Reviewer :
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What Is Methimazole and How Does It Work?

Methimazole is used to treat overactive thyroid (hyperthyroidism). It works by stopping the thyroid gland from making too much thyroid hormone.

  • Methimazole is available under the following different brand names: Northyx, and Tapazole.

What Are Dosages of Methimazole?

Dosages of Methimazole:

Adult and Pediatric Dosage Forms and Strengths

Tablet

  • 5 mg
  • 10 mg

Dosing Considerations – Should be Given as Follows:

Hyperthyroidism

Adult:

  • Mild: 15 mg/day orally divided every 8 hours initially
  • Moderate: 30-40 mg/day orally divided every 8 hours initially
  • Severe: 60 mg/day orally divided every 8 hours initially
  • Maintenance: 5-15 mg/day orally divided every 8 hours

Pediatric:

  • Initial: 0.4-0.7 mg/kg/day orally divided every 8 hours
  • Maintenance: 1/3-2/3 of initial orally dosage divided every 8 hours orally
  • Not to exceed 30 mg/day

Graves Disease

  • Adult: 10-20 mg/day orally; after euthyroidism is achieved, reduce dosage by 50% and administer for 12-18 months
  • Pediatric: 0.2-0.5 mg/kg/day orally; after euthyroidism is achieved, reduce dosage by 50% and administered for 1-2 years

Thyrotoxic Crisis

  • 20-30 mg every 6-12 hours for the short term, then reduce dosage to maintenance (5-15 mg/day) or reduce the frequency to every 12 hours or every 24 hours

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